Profile

Name

Hiroaki Ishida

Affiliation

Lavoratory of Drug Design and Medicinal Chemistry

Subjects

　

Official title

Senior Assistant professor

Degree

Ph.D.

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Papers

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• Original paper　2-cyanopyridine derivatives enable N-terminal cysteine bioconjugation and peptide bond cleavage of glutathione under aqueous and mild conditions.　Yano T, Yamada T*, Ishida H, Ohashi N, Itoh T*.　RSC Adv.　14　6542-6547.　2024　[Related links]
• Original paper　Covalent Modifier Discovery using Hydrogen/Deuterium Exchange–Mass Spectrometry.　Kojima H, Yanagi R, Higuchi E, Yoshizawa M, Shimodaira T, Kumagai M, Kyoya T, Sekine M, Egawa D, Ohashi N, Ishida H, Yamamoto K, Itoh T*.　J. Med. Chem.　66　4827–4839.　2023　[Related links]
• Original paper　Synthesis of triazolo[c]coumarins and differences in the fluorescence properties of their isomers.　Sekine M, Ishida H, Itoh T*.　Asian J. Org. Chem.　12　e202300013　2023　[Related links]
• Original paper　Oligoarginine-conjugated peptide foldamers inhibiting vitamin D receptor-mediated transcription.　Takyo M, Sato Y, Hirata N, Tsuchiya K, Ishida H, Kurohara T, Yanase Y, Ito T, Kanda Y, Yamamoto K, Misawa T*, Demizu Y*.　ACS Omega　7　46573–46582.　2022　[Related links]
• Original paper　Synthesis of Tetrahydrofuro[2,3-d]oxazoles and Oxazoles by Hypervalent Iodine (III) Promoted [2 + 2 + 1] Annulation.　Ishida H*, Homma S, Kasuga R, Yamamoto K, Itoh T*　Chem. Pharm. Bull.　70　192?194.　2022　[Related links]
• Original paper　Construction of 7-diethylaminocoumarins promoted by an electro-withdrawing group.　Yoshikawa C, Ishida H, Ohashi N, Kojima H, Itoh T.　Chem. Pharm. Bull.　69　608–611.　2021　[Related links]
• Original paper　Synthesis of a Coumarin-Based PPARγ Fluorescence Probe for Competitive Binding Assay.　Yoshikawa C, Ishida H, Ohashi N, Itoh T.　Int. J. Mol. Sci.　22　4034　2021　[Related links]
• Original paper　HNF4α Is a Covalent Bond-Forming Receptor.　Kanamori S, Ohashi N, Ishida H, Yamamoto K, Itoh T*.　J. Nutr. Sci. Vitaminol.　67　126–129　2021　[Related links]
• Original paper　Lithocholic Acid Derivatives as Potent Vitamin D Receptor Agonists.　Sasaki H, Masuno H, Kawasaki H, Yoshihara A, Numoto, N, Ito N, Ishida H, Yamamoto K, Hirata N, Kanda Y, Kawachi E, Kagechika H, and Tanatani A.　J. Med. Chem.　64　516?526.　2021　[Related links]
• Original paper　Incorporation of a coumarin unit by nucleophilic addition reaction into a PPARγ ligand.　Yoshikawa C, Ishida H, Itoh T.　Tetrahedron Lett.　61　151842　2020　[Related links]
• Original paper　Construction of a series of intermediates in the β-oxidation pathway from THA to EPA via DHA in free acid form.　Kanamori S, Ishida H, Yamamoto K, Itoh T.　Bioorg. Med. Chem.　26　4390–4401　2018　[Related links]
• Original paper　Vitamin D analogues with a p-hydroxyphenyl group at the C25 position: crystal structure of vitamin D receptor ligand-binding domain complexed with the ligand explains the mechanism underlying full antagonistic action.　Kato A, Yamao M, Hashihara Y, Ishida H, Itoh T, Yamamoto K.　J. Med. Chem.　60　8394-8406　2017　[Related links]
• Original paper　Three-Component Regioselective Synthesis of Tetrahydrofuro[2,3-d]oxazoles and their Efficient Conversion to Oxazoles.　Ohura A, Itoh T, Ishida H, Saito A, Yamamoto K.　Asian J. Org. Chem.　6　673-676.　2017　[Related links]
• [Original paper]　Gram scale synthesis of specialized pro-resolving mediator 17(S)-HDHA using lipoxygenase enhanced by water-soluble reducing agent TCEP.　Itoh T, Saito T, Yamamoto Y, Ishida H, Yamamoto K　Bioorganic & Medicinal Chemistry Letters　26　343-345　2016　
• [Original paper]　The First Asymmetric Total Synthesis of Lycoposerramine-R.　H. Ishida, S. Kimura, N. Kogure, M. Kitajima, and H. Takayama.　Organic & Biomolecular Chemistry　13　7762-7771　2015　
• [Original paper]　Total synthesis of (±)-lycoposerramine-R, a novel skeletal type of Lycopodium alkaloid.　H. Ishida, S. Kimura, N. Kogure, M. Kitajima, and H. Takayama.　Tetrahedron　71　51-56　2015　

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Conference, etc.

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• [Oral presentation]　新規骨格LycopodiumアルカロイドLycoposerramine-R の不斉全合成　石田寛明，木村真也，小暮紀行，北島満里子，高山廣光　第135年会日本薬学会　神戸　2015/03/25～2015/03/28
• [Oral presentation]　新規骨格LycopodiumアルカロイドLycoposerramine-R の不斉全合成研究　石田寛明，木村真也，小暮紀行，北島満里子，高山廣光　第40回反応と合成の進歩シンポジウム　仙台　2014/11/10～2014/11/11
• [Poster presentation]　新規骨格LycopodiumアルカロイドLycoposerramine-R の不斉全合成研究　石田寛明，木村真也，小暮紀行，北島満里子，高山廣光　第134年会日本薬学会　熊本　2014/03/27～2014/03/30
• [Oral presentation]　Study on Asymmetric Total Synthesis of Lycoposerramine-R, A Novel Skeletal Type of Lycopodium Alkaloids　石田寛明，木村真也，小暮紀行，北島満里子，高山廣光　Workshop on Chirality in Chiba University - 2nd Symposium　千葉　2014/01/31
• [Poster presentation]　新規骨格LycopodiumアルカロイドLycoposerramine-R の不斉全合成研究　石田寛明，木村真也，小暮紀行，北島満里子，高山廣光　第48回天然物化学談話会　大津　2013/07/03～2013/07/05
• [Poster presentation]　新規骨格LycopodiumアルカロイドLycoposerramine-R の不斉全合成研究　石田寛明，木村真也，小暮紀行，北島満里子，高山廣光　第133年会日本薬学会　横浜　2013/03/27～2013/03/30
• [Poster presentation]　新規骨格LycopodiumアルカロイドLycoposerramine-R の不斉全合成研究　石田寛明，木村真也，小暮紀行，北島満里子，高山廣光　第47回天然物化学談話会　阿蘇　2012/07/04～2012/07/06
• [Poster presentation]　10-Fluorocorynantheidine類の不斉全合成研究　石田　寛明,　小暮　紀行, 北島　満里子, 高山　廣光　第132年会日本薬学会　札幌　2012/03/28～2012/03/31

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